Friday, January 20, 2023

Oxidation of Fatty Acids (β-oxidation)

 Oxidation of Fatty Acids (β-oxidation)

Introduction

The process of successive β-oxidation was described by Knoop in 1905. In this process the oxidation takes place in the carbon atom at the β-position (third from the carboxyl group). This carbon atom is converted into a carboxyl (-COOH) group and the outer two-carbon atoms are split off. Thus a fatty acid with two-carbon atoms less is formed. That substance again undergoes β-oxidation and the process is repeated successively, Thus fatty acid oxidation takes place in a process known as alternate successive β-oxidation where two-carbon atoms are removed at a time as acetic acid, until a four-carbon atom residue is left as butyric acid. Butyric acid is oxidized in the β-position to form acetoacetic acid. Consequently, the original fatty acid molecule is converted into several molecules of acetic acid and one molecule of acetoacetic acid (ketone). Both of these compounds undergo final oxidation into CO, and H₂O in normal health.

Stages

Discovery of coenzyme A (HS-CoA) by Lipmann and acetyl coenzyme A or active acetate by Lynen and his colleagues has explained the process further. Coenzyme A has been found to be in large quantity in the liver. Coenzyme A is a dinucleotide and consists of 2-thiol-ethylamine and pantothenic acid linked with pyrophosphate and adenosine. Active acetate is an acetylated derivative of this coenzyme. The sulphur atom is linked to acetyl group. The neutral fat is hydrolyzed in the liver into long-chain fatty acids (Palmitic, Stearic and Oleic acids containing 16 or 18 carbon atoms) and glycerol.

The fatty acid radical undergoes successive oxidation in the liver and breaks down into smaller fragments in the following stages-

1. Stage of activation- Fatty acid is activated by thiokinase in presence of coenzyme A, ATP and Mg++ and activated fatty acid or coenzyme ester is formed. There are at least three kinases that catalyze the acylation of fatty acid. Acetic kinase shows a high specificity for acetic acid and slightly for propionic acid. A second kinase acts on acids C4-C12, optimum chain length being C8. The long-chain kinase (C8-C16) has little action on short-chain acids.

2. Stage of Dehydrogenation- The activated fatty acid is oxidized by the removal of two hydrogen atoms by acyl-CoA dehydrogenase along with a coenzyme derived from flavin adenine dinucleotide (FAD) and α-β-unsaturated activated fatty acid is produced. Just as in case of kinases, there are at least three dehydrogenases, viz., G, Y, and Y₂. C green-colored dehydrogenase which catalyses oxidation of C4-C8 acids, Y₁ is yellow, having optimal action on C8-C12 acids and Y₂ being m active on C8-C16 acids.

3.Stage of Hydration-Then a-ß-unsaturated fatty acid passes through process of hydration with the addition of H₂O under the influence of enoyl hydrase (crotonase) and β-hydroxy activated fatty acid is produced which undergoes dehydrogenation again.

4. Stage of Dehydrogenation-There is removal of two hydrogen atoms from ß-carbon atoms, and ß -keto activated fatty acid is produced. NAD acts as a hydrogen acceptor being converted into NADH2. This reaction is catalysed by ß-hydroxyacyl CoA dehydrogenase.

(V) Stage of thiolytic cleavage-β-keto activated fatty acid is cleavaged 3-carbon atom, by thiolase (8-ketothiolase) in presence of CoASH and thus two-carbon fragment as acetyl CoA is separated leaving activate fatty acid less by 2C. This process is repeated again and again and an acetyl CoA is separated off in each complete oxidation process till the fatty acid completely split into two-carbon fragments (acetyl CoA).

Even-carbon fatty acids, undergoing β-oxidation, even carbon fatty acids give rise to acetyl CoA whereas odd-carbon fatty acids also give rise to acetyl CoA and a molecule of propionyl CoA, the latter being formed from the 3 terminal carbon atoms from the methyl end of fatty acid.

Branched-chain fatty acids (e, isobutyric and isocaproic acids, etc.) are also split into acetyl CoA and propionyl CoA during their oxidation. The propionyl CoA converted to methyl malonyl CoA and finally isomerized to succinyl CoA. The succinyl CoA may be utilized for the synthesis of carbohydrate through pyruvic acid and porphyrin with glycine or may be oxidized through TCA cycle after being converted into succinic acid to supply energy as ATP. Acetyl CoA is oxidized in the TCA cycle and the coenzyme A thus set free after oxidation helps further fatty acid oxidation. If acetyl CoA is not properly oxidized, aceto-acetic acid is produced,

Fatty acid oxidation depends upon simultaneous oxidation of carbohydrate.

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